Splicing modulators act at the branch point adenosine binding pocket defined by the PHF5A-SF3b complex.
Nature Communications
Teng, Teng T; Tsai, Jennifer Hc JH; Puyang, Xiaoling X; Seiler, Michael M; Peng, Shouyong S; Prajapati, Sudeep S; Aird, Daniel D; Buonamici, Silvia S; Caleb, Benjamin B; Chan, Betty B; Corson, Laura L; Feala, Jacob J; Fekkes, Peter P; Gerard, Baudouin B; Karr, Craig C; Korpal, Manav M; Liu, Xiang X; T Lowe, Jason J; Mizui, Yoshiharu Y; Palacino, James J; Park, Eunice E; Smith, Peter G PG; Subramanian, Vanitha V; Wu, Zhenhua Jeremy ZJ; Zou, Jian J; Yu, Lihua L; Chicas, Agustin A; Warmuth, Markus M; Larsen, Nicholas N; Zhu, Ping P