Discovery of potent SOS1 inhibitors that block RAS activation via disruption of the RAS-SOS1 interaction.
Proceedings Of The National Academy Of Sciences Of The United States Of America
Hillig, Roman C RC; Sautier, Brice B; Schroeder, Jens J; Moosmayer, Dieter D; Hilpmann, André A; Stegmann, Christian M CM; Werbeck, Nicolas D ND; Briem, Hans H; Boemer, Ulf U; Weiske, Joerg J; Badock, Volker V; Mastouri, Julia J; Petersen, Kirstin K; Siemeister, Gerhard G; Kahmann, Jan D JD; Wegener, Dennis D; Böhnke, Niels N; Eis, Knut K; Graham, Keith K; Wortmann, Lars L; von Nussbaum, Franz F; Bader, Benjamin B
Contact inhibition modulates intracellular levels of miR-223 in a p27kip1-dependent manner.
Oncotarget
Armenia, Joshua J; Fabris, Linda L; Lovat, Francesca F; Berton, Stefania S; Segatto, Ilenia I; D'Andrea, Sara S; Ivan, Cristina C; Cascione, Luciano L; Calin, George A GA; Croce, Carlo M CM; Colombatti, Alfonso A; Vecchione, Andrea A; Belletti, Barbara B; Baldassarre, Gustavo G