Targeting oncogenic KRasG13C with nucleotide-based covalent inhibitors.
Elife
Goebel, Lisa L; Kirschner, Tonia T; Koska, Sandra S; Rai, Amrita A; Janning, Petra P; Maffini, Stefano S; Vatheuer, Helge H; Czodrowski, Paul P; Goody, Roger S RS; Müller, Matthias P MP; Rauh, Daniel D
Oncogenic KRAS G12C: Kinetic and redox characterization of covalent inhibition.
The Journal Of Biological Chemistry
Huynh, Minh V MV; Parsonage, Derek D; Forshaw, Tom E TE; Chirasani, Venkat R VR; Hobbs, G Aaron GA; Wu, Hanzhi H; Lee, Jingyun J; Furdui, Cristina M CM; Poole, Leslie B LB; Campbell, Sharon L SL
Computationally Empowered Workflow Identifies Novel Covalent Allosteric Binders for KRASG12C.
Chemmedchem
Mortier, Jérémie J; Friberg, Anders A; Badock, Volker V; Moosmayer, Dieter D; Schroeder, Jens J; Steigemann, Patrick P; Siegel, Franziska F; Gradl, Stefan S; Bauser, Marcus M; Hillig, Roman C RC; Briem, Hans H; Eis, Knut K; Bader, Benjamin B; Nguyen, Duy D; Christ, Clara D CD
Proceedings Of The National Academy Of Sciences Of The United States Of America
Kessler, Dirk D; Gmachl, Michael M; Mantoulidis, Andreas A; Martin, Laetitia J LJ; Zoephel, Andreas A; Mayer, Moriz M; Gollner, Andreas A; Covini, David D; Fischer, Silke S; Gerstberger, Thomas T; Gmaschitz, Teresa T; Goodwin, Craig C; Greb, Peter P; Häring, Daniela D; Hela, Wolfgang W; Hoffmann, Johann J; Karolyi-Oezguer, Jale J; Knesl, Petr P; Kornigg, Stefan S; Koegl, Manfred M; Kousek, Roland R; Lamarre, Lyne L; Moser, Franziska F; Munico-Martinez, Silvia S; Peinsipp, Christoph C; Phan, Jason J; Rinnenthal, Jörg J; Sai, Jiqing J; Salamon, Christian C; Scherbantin, Yvonne Y; Schipany, Katharina K; Schnitzer, Renate R; Schrenk, Andreas A; Sharps, Bernadette B; Siszler, Gabriella G; Sun, Qi Q; Waterson, Alex A; Wolkerstorfer, Bernhard B; Zeeb, Markus M; Pearson, Mark M; Fesik, Stephen W SW; McConnell, Darryl B DB