ASN007 is a selective ERK1/2 inhibitor with preferential activity against RAS-and RAF-mutant tumors.
Cell Reports. Medicine
Portelinha, Ana A; Thompson, Scott S; Smith, Roger A RA; Da Silva Ferreira, Mariana M; Asgari, Zahra Z; Knezevic, Andrea A; Seshan, Venkatraman V; de Stanchina, Elisa E; Gupta, Sandeep S; Denis, Louis L; Younes, Anas A; Reddy, Sanjeeva S