The SMARCA2/4 ATPase Domain Surpasses the Bromodomain as a Drug Target in SWI/SNF-Mutant Cancers: Insights from cDNA Rescue and PFI-3 Inhibitor Studies.
Cancer Research
Vangamudi, Bhavatarini B; Paul, Thomas A TA; Shah, Parantu K PK; Kost-Alimova, Maria M; Nottebaum, Lisa L; Shi, Xi X; Zhan, Yanai Y; Leo, Elisabetta E; Mahadeshwar, Harshad S HS; Protopopov, Alexei A; Futreal, Andrew A; Tieu, Trang N TN; Peoples, Mike M; Heffernan, Timothy P TP; Marszalek, Joseph R JR; Toniatti, Carlo C; Petrocchi, Alessia A; Verhelle, Dominique D; Owen, Dafydd R DR; Draetta, Giulio G; Jones, Philip P; Palmer, Wylie S WS; Sharma, Shikhar S; Andersen, Jannik N JN