Lucanthone and its derivative hycanthone inhibit apurinic endonuclease-1 (APE1) by direct protein binding.
Plos One
Naidu, Mamta D MD; Agarwal, Rakhi R; Pena, Louis A LA; Cunha, Luis L; Mezei, Mihaly M; Shen, Min M; Wilson, David M DM; Liu, Yuan Y; Sanchez, Zina Z; Chaudhary, Pankaj P; Wilson, Samuel H SH; Waring, Michael J MJ