DFG-out mode of inhibition by an irreversible type-1 inhibitor capable of overcoming gate-keeper mutations in FGF receptors.
Acs Chemical Biology
Huang, Zhifeng Z; Tan, Li L; Wang, Huiyan H; Liu, Yang Y; Blais, Steven S; Deng, Jingjing J; Neubert, Thomas A TA; Gray, Nathanael S NS; Li, Xiaokun X; Mohammadi, Moosa M