Design and Synthesis of Type-IV Inhibitors of BRAF Kinase That Block Dimerization and Overcome Paradoxical MEK/ERK Activation.
Journal Of Medicinal Chemistry
Beneker, Chad M CM; Rovoli, Magdalini M; Kontopidis, George G; Röring, Michael M; Galda, Simeon S; Braun, Sandra S; Brummer, Tilman T; McInnes, Campbell C
The Origins and Vulnerabilities of Two Transmissible Cancers in Tasmanian Devils.
Cancer Cell
Stammnitz, Maximilian R MR; Coorens, Tim H H THH; Gori, Kevin C KC; Hayes, Dane D; Fu, Beiyuan B; Wang, Jinhong J; Martin-Herranz, Daniel E DE; Alexandrov, Ludmil B LB; Baez-Ortega, Adrian A; Barthorpe, Syd S; Beck, Alexandra A; Giordano, Francesca F; Knowles, Graeme W GW; Kwon, Young Mi YM; Hall, George G; Price, Stacey S; Pye, Ruth J RJ; Tubio, Jose M C JMC; Siddle, Hannah V T HVT; Sohal, Sukhwinder Singh SS; Woods, Gregory M GM; McDermott, Ultan U; Yang, Fengtang F; Garnett, Mathew J MJ; Ning, Zemin Z; Murchison, Elizabeth P EP
Systematic identification of genomic markers of drug sensitivity in cancer cells.
Nature
Garnett, Mathew J MJ; Edelman, Elena J EJ; Heidorn, Sonja J SJ; Greenman, Chris D CD; Dastur, Anahita A; Lau, King Wai KW; Greninger, Patricia P; Thompson, I Richard IR; Luo, Xi X; Soares, Jorge J; Liu, Qingsong Q; Iorio, Francesco F; Surdez, Didier D; Chen, Li L; Milano, Randy J RJ; Bignell, Graham R GR; Tam, Ah T AT; Davies, Helen H; Stevenson, Jesse A JA; Barthorpe, Syd S; Lutz, Stephen R SR; Kogera, Fiona F; Lawrence, Karl K; McLaren-Douglas, Anne A; Mitropoulos, Xeni X; Mironenko, Tatiana T; Thi, Helen H; Richardson, Laura L; Zhou, Wenjun W; Jewitt, Frances F; Zhang, Tinghu T; O'Brien, Patrick P; Boisvert, Jessica L JL; Price, Stacey S; Hur, Wooyoung W; Yang, Wanjuan W; Deng, Xianming X; Butler, Adam A; Choi, Hwan Geun HG; Chang, Jae Won JW; Baselga, Jose J; Stamenkovic, Ivan I; Engelman, Jeffrey A JA; Sharma, Sreenath V SV; Delattre, Olivier O; Saez-Rodriguez, Julio J; Gray, Nathanael S NS; Settleman, Jeffrey J; Futreal, P Andrew PA; Haber, Daniel A DA; Stratton, Michael R MR; Ramaswamy, Sridhar S; McDermott, Ultan U; Benes, Cyril H CH