Drug trapping in hERG K+ channels: (not) a matter of drug size?
Medchemcomm
Linder, Tobias T; Bernsteiner, Harald H; Saxena, Priyanka P; Bauer, Florian F; Erker, Thomas T; Timin, Eugen E; Hering, Steffen S; Stary-Weinzinger, Anna A
Transfer of rolf S3-S4 linker to HERG eliminates activation gating but spares inactivation.
Biophysical Journal
Choveau, Frank S FS; El Harchi, Aziza A; Rodriguez, Nicolas N; Louérat-Oriou, Bénédicte B; Baró, Isabelle I; Demolombe, Sophie S; Charpentier, Flavien F; Loussouarn, Gildas G