Chaperones as thermodynamic sensors of drug-target interactions reveal kinase inhibitor specificities in living cells.
Nature Biotechnology
Taipale, Mikko M; Krykbaeva, Irina I; Whitesell, Luke L; Santagata, Sandro S; Zhang, Jianming J; Liu, Qingsong Q; Gray, Nathanael S NS; Lindquist, Susan S
Targeting Bcr-Abl by combining allosteric with ATP-binding-site inhibitors.
Nature
Zhang, Jianming J; Adrián, Francisco J FJ; Jahnke, Wolfgang W; Cowan-Jacob, Sandra W SW; Li, Allen G AG; Iacob, Roxana E RE; Sim, Taebo T; Powers, John J; Dierks, Christine C; Sun, Fangxian F; Guo, Gui-Rong GR; Ding, Qiang Q; Okram, Barun B; Choi, Yongmun Y; Wojciechowski, Amy A; Deng, Xianming X; Liu, Guoxun G; Fendrich, Gabriele G; Strauss, André A; Vajpai, Navratna N; Grzesiek, Stephan S; Tuntland, Tove T; Liu, Yi Y; Bursulaya, Badry B; Azam, Mohammad M; Manley, Paul W PW; Engen, John R JR; Daley, George Q GQ; Warmuth, Markus M; Gray, Nathanael S NS