Identification of Novel Small Molecule Ligands for JAK2 Pseudokinase Domain.
Pharmaceuticals (Basel, Switzerland)
Virtanen, Anniina T AT; Haikarainen, Teemu T; Sampathkumar, Parthasarathy P; Palmroth, Maaria M; Liukkonen, Sanna S; Liu, Jianping J; Nekhotiaeva, Natalia N; Hubbard, Stevan R SR; Silvennoinen, Olli O
Selective Janus Kinase 2 (JAK2) Pseudokinase Ligands with a Diaminotriazole Core.
Journal Of Medicinal Chemistry
Liosi, Maria-Elena ME; Krimmer, Stefan G SG; Newton, Ana S AS; Dawson, Thomas K TK; Puleo, David E DE; Cutrona, Kara J KJ; Suzuki, Yoshihisa Y; Schlessinger, Joseph J; Jorgensen, William L WL
Uncoupling JAK2 V617F activation from cytokine-induced signalling by modulation of JH2 αC helix.
The Biochemical Journal
Leroy, Emilie E; Dusa, Alexandra A; Colau, Didier D; Motamedi, Amir A; Cahu, Xavier X; Mouton, Céline C; Huang, Lily J LJ; Shiau, Andrew K AK; Constantinescu, Stefan N SN