Incorporation of Agouti-Related Protein (AgRP) Human Single Nucleotide Polymorphisms (SNPs) in the AgRP-Derived Macrocyclic Scaffold c[Pro-Arg-Phe-Phe-Asn-Ala-Phe-dPro] Decreases Melanocortin-4 Receptor Antagonist Potency and Results in the Discovery of Melanocortin-5 Receptor Antagonists.
Journal Of Medicinal Chemistry
Koerperich, Zoe M ZM; Ericson, Mark D MD; Freeman, Katie T KT; Speth, Robert C RC; Pogozheva, Irina D ID; Mosberg, Henry I HI; Haskell-Luevano, Carrie C
Publication Date: 2020-03-12
Variant appearance in text: AGRP: R111C; rs1012110755