Structure-activity relationships of peptides incorporating a bioactive reverse-turn heterocycle at the melanocortin receptors: identification of a 5800-fold mouse melanocortin-3 receptor (mMC3R) selective antagonist/partial agonist versus the mouse melanocortin-4 receptor (mMC4R).
Journal Of Medicinal Chemistry
Singh, Anamika A; Dirain, Marvin M; Witek, Rachel R; Rocca, James R JR; Edison, Arthur S AS; Haskell-Luevano, Carrie C