JAK-STAT signaling in inflammatory breast cancer enables chemotherapy-resistant cell states.
Cancer Research
Stevens, Laura E LE; Peluffo, Guillermo G; Qiu, Xintao X; Temko, Daniel D; Fassl, Anne A; Li, Zheqi Z; Trinh, Anne A; Seehawer, Marco M; Jovanovic, Bojana B; Aleckovic, Masa M; Wilde, Callahan M CM; Geck, Renee C RC; Shu, Shaokun S; Kingston, Natalie L NL; Harper, Nicholas W NW; Almendro, Vanessa V; Pyke, Alanna L AL; Egri, Shawn B SB; Papanastasiou, Malvina M; Clement, Kendell K; Zhou, Ningxuan N; Walker, Sarah S; Salas, Jacqueline J; Park, So Yeon SY; Frank, David A DA; Meissner, Alexander A; Jaffe, Jacob D JD; Sicinski, Piotr P; Toker, Alex A; Michor, Franziska F; Long, Henry W HW; Overmoyer, Beth A BA; Polyak, Kornelia K
Maintaining protein stability of ∆Np63 via USP28 is required by squamous cancer cells.
Embo Molecular Medicine
Prieto-Garcia, Cristian C; Hartmann, Oliver O; Reissland, Michaela M; Braun, Fabian F; Fischer, Thomas T; Walz, Susanne S; Schülein-Völk, Christina C; Eilers, Ursula U; Ade, Carsten P CP; Calzado, Marco A MA; Orian, Amir A; Maric, Hans M HM; Münch, Christian C; Rosenfeldt, Mathias M; Eilers, Martin M; Diefenbacher, Markus E ME
Mutational processes shape the landscape of TP53 mutations in human cancer.
Nature Genetics
Giacomelli, Andrew O AO; Yang, Xiaoping X; Lintner, Robert E RE; McFarland, James M JM; Duby, Marc M; Kim, Jaegil J; Howard, Thomas P TP; Takeda, David Y DY; Ly, Seav Huong SH; Kim, Eejung E; Gannon, Hugh S HS; Hurhula, Brian B; Sharpe, Ted T; Goodale, Amy A; Fritchman, Briana B; Steelman, Scott S; Vazquez, Francisca F; Tsherniak, Aviad A; Aguirre, Andrew J AJ; Doench, John G JG; Piccioni, Federica F; Roberts, Charles W M CWM; Meyerson, Matthew M; Getz, Gad G; Johannessen, Cory M CM; Root, David E DE; Hahn, William C WC
Capzimin is a potent and specific inhibitor of proteasome isopeptidase Rpn11.
Nature Chemical Biology
Li, Jing J; Yakushi, Tanya T; Parlati, Francesco F; Mackinnon, Andrew L AL; Perez, Christian C; Ma, Yuyong Y; Carter, Kyle P KP; Colayco, Sharon S; Magnuson, Gavin G; Brown, Brock B; Nguyen, Kevin K; Vasile, Stefan S; Suyama, Eigo E; Smith, Layton H LH; Sergienko, Eduard E; Pinkerton, Anthony B AB; Chung, Thomas D Y TDY; Palmer, Amy E AE; Pass, Ian I; Hess, Sonja S; Cohen, Seth M SM; Deshaies, Raymond J RJ
Aurora kinases in childhood acute leukemia: the promise of aurora B as therapeutic target.
Leukemia
Hartsink-Segers, S A SA; Zwaan, C M CM; Exalto, C C; Luijendijk, M W J MW; Calvert, V S VS; Petricoin, E F EF; Evans, W E WE; Reinhardt, D D; de Haas, V V; Hedtjärn, M M; Hansen, B R BR; Koch, T T; Caron, H N HN; Pieters, R R; Den Boer, M L ML