Biological Profiling Enables Rapid Mechanistic Classification of Phenotypic Screening Hits and Identification of KatG Activation-Dependent Pyridine Carboxamide Prodrugs With Activity Against Mycobacterium tuberculosis.
Frontiers In Cellular And Infection Microbiology
Chengalroyen, Melissa D MD; Jordaan, Audrey A; Seldon, Ronnett R; Ioerger, Thomas T; Franzblau, Scott G SG; Nasr, Mohamed M; Warner, Digby F DF; Mizrahi, Valerie V
Determinants of the Inhibition of DprE1 and CYP2C9 by Antitubercular Thiophenes.
Angewandte Chemie (International Ed. In English)
Liu, Renhe R; Lyu, Xiaoxuan X; Batt, Sarah M SM; Hsu, Mei-Hui MH; Harbut, Michael B MB; Vilchèze, Catherine C; Cheng, Bo B; Ajayi, Kehinde K; Yang, Baiyuan B; Yang, Yun Y; Guo, Hui H; Lin, Changyou C; Gan, Fei F; Wang, Chen C; Franzblau, Scott G SG; Jacobs, William R WR; Besra, Gurdyal S GS; Johnson, Eric F EF; Petrassi, Mike M; Chatterjee, Arnab K AK; Fütterer, Klaus K; Wang, Feng F
Identification of a small molecule with activity against drug-resistant and persistent tuberculosis.
Proceedings Of The National Academy Of Sciences Of The United States Of America
Wang, Feng F; Sambandan, Dhinakaran D; Halder, Rajkumar R; Wang, Jianing J; Batt, Sarah M SM; Weinrick, Brian B; Ahmad, Insha I; Yang, Pengyu P; Zhang, Yong Y; Kim, John J; Hassani, Morad M; Huszar, Stanislav S; Trefzer, Claudia C; Ma, Zhenkun Z; Kaneko, Takushi T; Mdluli, Khisi E KE; Franzblau, Scott S; Chatterjee, Arnab K AK; Johnsson, Kai K; Johnson, Kai K; Mikusova, Katarina K; Besra, Gurdyal S GS; Fütterer, Klaus K; Robbins, Scott H SH; Barnes, S Whitney SW; Walker, John R JR; Jacobs, William R WR; Schultz, Peter G PG