A highly sensitive cell-based luciferase assay for high-throughput automated screening of SARS-CoV-2 nsp5/3CLpro inhibitors.
Antiviral Research
Chen, K Y KY; Krischuns, T T; Varga, L Ortega LO; Harigua-Souiai, E E; Paisant, S S; Zettor, A A; Chiaravalli, J J; Delpal, A A; Courtney, D D; O'Brien, A A; Baker, S C SC; Decroly, E E; Isel, C C; Agou, F F; Jacob, Y Y; Blondel, A A; Naffakh, N N
A highly sensitive cell-based luciferase assay for high-throughput automated screening of SARS-CoV-2 nsp5/3CLpro inhibitors.
Biorxiv : The Preprint Server For Biology
Chen, K Y KY; Krischuns, T T; Ortega Varga, L L; Harigua-Souiai, E E; Paisant, S S; Zettor, A A; Chiaravalli, J J; Courtney, D D; O'Brien, A A; Baker, S C SC; Isel, C C; Agou, F F; Jacob, Y Y; Blondel, A A; Naffakh, N N
Large-Scale Recombinant Production of the SARS-CoV-2 Proteome for High-Throughput and Structural Biology Applications.
Frontiers In Molecular Biosciences
Altincekic, Nadide N; Korn, Sophie Marianne SM; Qureshi, Nusrat Shahin NS; Dujardin, Marie M; Ninot-Pedrosa, Martí M; Abele, Rupert R; Abi Saad, Marie Jose MJ; Alfano, Caterina C; Almeida, Fabio C L FCL; Alshamleh, Islam I; de Amorim, Gisele Cardoso GC; Anderson, Thomas K TK; Anobom, Cristiane D CD; Anorma, Chelsea C; Bains, Jasleen Kaur JK; Bax, Adriaan A; Blackledge, Martin M; Blechar, Julius J; Böckmann, Anja A; Brigandat, Louis L; Bula, Anna A; Bütikofer, Matthias M; Camacho-Zarco, Aldo R AR; Carlomagno, Teresa T; Caruso, Icaro Putinhon IP; Ceylan, Betül B; Chaikuad, Apirat A; Chu, Feixia F; Cole, Laura L; Crosby, Marquise G MG; de Jesus, Vanessa V; Dhamotharan, Karthikeyan K; Felli, Isabella C IC; Ferner, Jan J; Fleischmann, Yanick Y; Fogeron, Marie-Laure ML; Fourkiotis, Nikolaos K NK; Fuks, Christin C; Fürtig, Boris B; Gallo, Angelo A; Gande, Santosh L SL; Gerez, Juan Atilio JA; Ghosh, Dhiman D; Gomes-Neto, Francisco F; Gorbatyuk, Oksana O; Guseva, Serafima S; Hacker, Carolin C; Häfner, Sabine S; Hao, Bing B; Hargittay, Bruno B; Henzler-Wildman, K K; Hoch, Jeffrey C JC; Hohmann, Katharina F KF; Hutchison, Marie T MT; Jaudzems, Kristaps K; Jović, Katarina K; Kaderli, Janina J; Kalniņš, Gints G; Kaņepe, Iveta I; Kirchdoerfer, Robert N RN; Kirkpatrick, John J; Knapp, Stefan S; Krishnathas, Robin R; Kutz, Felicitas F; Zur Lage, Susanne S; Lambertz, Roderick R; Lang, Andras A; Laurents, Douglas D; Lecoq, Lauriane L; Linhard, Verena V; Löhr, Frank F; Malki, Anas A; Bessa, Luiza Mamigonian LM; Martin, Rachel W RW; Matzel, Tobias T; Maurin, Damien D; McNutt, Seth W SW; Mebus-Antunes, Nathane Cunha NC; Meier, Beat H BH; Meiser, Nathalie N; Mompeán, Miguel M; Monaca, Elisa E; Montserret, Roland R; Mariño Perez, Laura L; Moser, Celine C; Muhle-Goll, Claudia C; Neves-Martins, Thais Cristtina TC; Ni, Xiamonin X; Norton-Baker, Brenna B; Pierattelli, Roberta R; Pontoriero, Letizia L; Pustovalova, Yulia Y; Ohlenschläger, Oliver O; Orts, Julien J; Da Poian, Andrea T AT; Pyper, Dennis J DJ; Richter, Christian C; Riek, Roland R; Rienstra, Chad M CM; Robertson, Angus A; Pinheiro, Anderson S AS; Sabbatella, Raffaele R; Salvi, Nicola N; Saxena, Krishna K; Schulte, Linda L; Schiavina, Marco M; Schwalbe, Harald H; Silber, Mara M; Almeida, Marcius da Silva MDS; Sprague-Piercy, Marc A MA; Spyroulias, Georgios A GA; Sreeramulu, Sridhar S; Tants, Jan-Niklas JN; Tārs, Kaspars K; Torres, Felix F; Töws, Sabrina S; Treviño, Miguel Á MÁ; Trucks, Sven S; Tsika, Aikaterini C AC; Varga, Krisztina K; Wang, Ying Y; Weber, Marco E ME; Weigand, Julia E JE; Wiedemann, Christoph C; Wirmer-Bartoschek, Julia J; Wirtz Martin, Maria Alexandra MA; Zehnder, Johannes J; Hengesbach, Martin M; Schlundt, Andreas A
6-phenylpyrrolocytosine as a fluorescent probe to examine nucleotide flipping catalyzed by a DNA repair protein.
Biopolymers
Kotandeniya, Delshanee D; Rogers, Melanie S MS; Fernandez, Jenna J; Kanugula, Sreenivas S; Hudson, Robert H E RHE; Rodriguez, Freddys F; Lipscomb, John D JD; Tretyakova, Natalia N
Disulfiram is a direct and potent inhibitor of human O6-methylguanine-DNA methyltransferase (MGMT) in brain tumor cells and mouse brain and markedly increases the alkylating DNA damage.
Carcinogenesis
Paranjpe, Ameya A; Zhang, Ruiwen R; Ali-Osman, Francis F; Bobustuc, George C GC; Srivenugopal, Kalkunte S KS