Publications:

Computer-Aided Ligand Discovery for Estrogen Receptor Alpha.

International Journal Of Molecular Sciences

Bafna, Divya D; Ban, Fuqiang F; Rennie, Paul S PS; Singh, Kriti K; Cherkasov, Artem A

Publication Date: 2020-06-12

Variant appearance in text: ESR1: L372S

PubMed Link: 32545494

Variant Present in the following documents:

• Main text
• ijms-21-04193.pdf

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The SERM/SERD bazedoxifene disrupts ESR1 helix 12 to overcome acquired hormone resistance in breast cancer cells.

Elife

Fanning, Sean W SW; Jeselsohn, Rinath R; Dharmarajan, Venkatasubramanian V; Mayne, Christopher G CG; Karimi, Mostafa M; Buchwalter, Gilles G; Houtman, René R; Toy, Weiyi W; Fowler, Colin E CE; Han, Ross R; Lainé, Muriel M; Carlson, Kathryn E KE; Martin, Teresa A TA; Nowak, Jason J; Nwachukwu, Jerome C JC; Hosfield, David J DJ; Chandarlapaty, Sarat S; Tajkhorshid, Emad E; Nettles, Kendall W KW; Griffin, Patrick R PR; Shen, Yang Y; Katzenellenbogen, John A JA; Brown, Myles M; Greene, Geoffrey L GL

Publication Date: 2018-11-29

Variant appearance in text: ESR1: L372S

PubMed Link: 30489256

Variant Present in the following documents:

• Main text
• elife-37161.pdf

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Structural and Molecular Mechanisms of Cytokine-Mediated Endocrine Resistance in Human Breast Cancer Cells.

Molecular Cell

Stender, Joshua D JD; Nwachukwu, Jerome C JC; Kastrati, Irida I; Kim, Yohan Y; Strid, Tobias T; Yakir, Maayan M; Srinivasan, Sathish S; Nowak, Jason J; Izard, Tina T; Rangarajan, Erumbi S ES; Carlson, Kathryn E KE; Katzenellenbogen, John A JA; Yao, Xin-Qiu XQ; Grant, Barry J BJ; Leong, Hon S HS; Lin, Chin-Yo CY; Frasor, Jonna J; Nettles, Kendall W KW; Glass, Christopher K CK

Publication Date: 2017-03-16

Variant appearance in text: ESR1: Leu372Ser

PubMed Link: 28306507

Variant Present in the following documents:

• Main text

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